Buparlisib (BKM120), 50mg

Buparlisib (BKM120), 50mg

Buparlisib (BKM120), 10mM/1mL

Buparlisib (BKM120), 10mM/1mL

Buparlisib (BKM120), 1g

25.770,64 RON
SKU
SKM_S2247_1g

Buparlisib (BKM120, NVP-BKM120) is a selective PI3Kinhibitor of p110α/β/δ/γwith IC50of 52 nM/166 nM/116 nM/262 nM in cell-free assays, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4Kβ. Buparlisib induces apoptosis. Phase 2.

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Description

Buparlisib (BKM120, NVP-BKM120) is a selective PI3Kinhibitor of p110α/β/δ/γwith IC50of 52 nM/166 nM/116 nM/262 nM in cell-free assays, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4Kβ. Buparlisib induces apoptosis. Phase 2.