Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR)and α3β4 nAChRwith EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRswith EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation.
Price | 1.856,00 RON (preturile sunt fara TVA) |
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Description |
Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR)and α3β4 nAChRwith EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRswith EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation. |