Samuraciclib (ICEC0942) hydrochloride, 2mg

Samuraciclib (ICEC0942) hydrochloride, 2mg

Samuraciclib (ICEC0942) hydrochloride, 25mg

Samuraciclib (ICEC0942) hydrochloride, 25mg

Samuraciclib (ICEC0942) hydrochloride, 5mg

2.528,75 RON
SKU
SKM_S8722_5mg

Samuraciclib (ICEC0942) hydrochloride is a new, orally bioavailable CDK7inhibitor with an IC50 of 40nM. The IC50 values for CDK1, CDK2, CDK5 and CDK9 were 45-, 15-, 230- and 30-fold higher. ICEC0942 (CT7001) promotes cell cycle arrest and apoptosis.

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Description

Samuraciclib (ICEC0942) hydrochloride is a new, orally bioavailable CDK7inhibitor with an IC50 of 40nM. The IC50 values for CDK1, CDK2, CDK5 and CDK9 were 45-, 15-, 230- and 30-fold higher. ICEC0942 (CT7001) promotes cell cycle arrest and apoptosis.