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Romanian
Romanian
English|
Rolapitant (SCH-619734) is a selective and competitive antagonist of human substance P/NK1receptors with antiemetic activity. It has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold, as well as preferential affinity for human, guinea pig, gerbil and monkey NK1 receptors over rat, mouse and rabbit.
| Price | 5.442,00 RON (preturile sunt fara TVA) |
|---|---|
| Description |
Rolapitant (SCH-619734) is a selective and competitive antagonist of human substance P/NK1receptors with antiemetic activity. It has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold, as well as preferential affinity for human, guinea pig, gerbil and monkey NK1 receptors over rat, mouse and rabbit. |
