Ricolinostat (ACY-1215) , 50mg

Ricolinostat (ACY-1215) , 50mg

Ricolinostat (ACY-1215) , 10mM/1mL

Ricolinostat (ACY-1215) , 10mM/1mL

Ricolinostat (ACY-1215) , 1g

19.467,21 RON
SKU
SKM_S8001_1g

Ricolinostat (ACY-1215, Rocilinostat) is a selective HDAC6inhibitor with IC50of 5 nM in a cell-free assay. It is >10-fold more selective for HDAC6 than HDAC1/2/3 (class I HDACs) with slight activity against HDAC8, minimal activity against HDAC4/5/7/9/11, Sirtuin1, and Sirtuin2. Ricolinostat (ACY-1215) suppresses cell proliferation and promotes apoptosis. Phase 2.

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Description

Ricolinostat (ACY-1215, Rocilinostat) is a selective HDAC6inhibitor with IC50of 5 nM in a cell-free assay. It is >10-fold more selective for HDAC6 than HDAC1/2/3 (class I HDACs) with slight activity against HDAC8, minimal activity against HDAC4/5/7/9/11, Sirtuin1, and Sirtuin2. Ricolinostat (ACY-1215) suppresses cell proliferation and promotes apoptosis. Phase 2.