Raltegravir, 1g

Raltegravir, 1g

Pyrimethamine, 1g

Pyrimethamine, 1g

Raltegravir, 10mM/1mL

1.586,27 RON
SKU
SKM_S2005_10mM/1mL

Raltegravir is a potent integrase (IN)inhibitor for WT and S217Q PFV IN with IC50 of 90 nM and 40 nM in cell-free assays, respectively. It shows greater than 1000-fold selectivity for HIV-1 IN over several related Mg2+-dependent enzyme such as HCV polymerase, HIV reverse transcriptase, HIV RNaseH and human α-, β-, γ-polymerases.

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Description

Raltegravir is a potent integrase (IN)inhibitor for WT and S217Q PFV IN with IC50 of 90 nM and 40 nM in cell-free assays, respectively. It shows greater than 1000-fold selectivity for HIV-1 IN over several related Mg2+-dependent enzyme such as HCV polymerase, HIV reverse transcriptase, HIV RNaseH and human α-, β-, γ-polymerases.