Limba
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MK-2461 is a potent, multi-targeted inhibitor for c-Met(WT/mutants)with IC50of 0.4-2.5 nM, less potent to Ron, Flt1; 8- to 30-fold greater selectivity of c-Met targets versus FGFR1, FGFR2, FGFR3, PDGFRβ, KDR, Flt3, Flt4, TrkA, and TrkB. Phase 1/2.
Price | 1.658,00 RON (preturile sunt fara TVA) |
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Description |
MK-2461 is a potent, multi-targeted inhibitor for c-Met(WT/mutants)with IC50of 0.4-2.5 nM, less potent to Ron, Flt1; 8- to 30-fold greater selectivity of c-Met targets versus FGFR1, FGFR2, FGFR3, PDGFRβ, KDR, Flt3, Flt4, TrkA, and TrkB. Phase 1/2. |