Ribociclib succinate, 10mM/1mL

Ribociclib succinate, 10mM/1mL

Lesinurad sodium, 25mg

Lesinurad sodium, 25mg

Lesinurad sodium, 5mg

860,37 RON
SKU
SKM_S5189_5mg

Lesinurad (Selexipag, RDEA-594) sodium (Zurampic) is a selective uric acid reabsorptioninhibitor (SURI) under investigation for treatment of gout. Lesinurad sodium inhibits the uric acid transporter URAT1and Kidney transporter OATwith IC50/Km of 4.3 μM/0.85 μM and 3.5 μM/2 μM for OAT1 and OAT3, respectively.

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Description

Lesinurad (Selexipag, RDEA-594) sodium (Zurampic) is a selective uric acid reabsorptioninhibitor (SURI) under investigation for treatment of gout. Lesinurad sodium inhibits the uric acid transporter URAT1and Kidney transporter OATwith IC50/Km of 4.3 μM/0.85 μM and 3.5 μM/2 μM for OAT1 and OAT3, respectively.