Fostamatinib (R788) disodium, 50mg

Fostamatinib (R788) disodium, 50mg

PIK-293, 5mg

PIK-293, 5mg

Fostamatinib (R788) disodium, 250mg

12.909,12 RON
SKU
SKM_S2206_250mg

Fostamatinib disodium (R788, Tamatinib Fosdium), a prodrug of the active metabolite R406, is a Sykinhibitor with IC50of 41 nM in a cell-free assay, strongly inhibits Syk but not Lyn, 5-fold less potent to Flt3. Phase 3.

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Description

Fostamatinib disodium (R788, Tamatinib Fosdium), a prodrug of the active metabolite R406, is a Sykinhibitor with IC50of 41 nM in a cell-free assay, strongly inhibits Syk but not Lyn, 5-fold less potent to Flt3. Phase 3.