Cirtuvivint, 5mg

Cirtuvivint, 5mg

SR 2640 hydrochloride, 5mg

SR 2640 hydrochloride, 5mg

Cirtuvivint, 25mg

9.688,98 RON
SKU
SKM_E2668_25mg

Cirtuvivint (SM08502) is a potent and orally active inhibitor of CDC-like kinase (CLK)and a DYRK(dual-specificity tyrosine kinase) that targets mRNA splicing and is optimized for Wnt pathway inhibition. Cirtuvivint inhibits serine and arginine-rich splicing factor (SRSF) phosphorylation and disrupts spliceosome activity. Cirtuvivint can be used for solid tumor research.

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Description

Cirtuvivint (SM08502) is a potent and orally active inhibitor of CDC-like kinase (CLK)and a DYRK(dual-specificity tyrosine kinase) that targets mRNA splicing and is optimized for Wnt pathway inhibition. Cirtuvivint inhibits serine and arginine-rich splicing factor (SRSF) phosphorylation and disrupts spliceosome activity. Cirtuvivint can be used for solid tumor research.