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Romanian
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Brilanestrant (GDC-0810), 5mg
1.180,48 RON
SKU
SKM_S7855_5mg
Brilanestrant (GDC-0810, ARN-810） is a potent ER-αbinder (ER-α, IC50 = 6.1 nM; ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 breast cancer cell viability (IC50 = 2.5 nM) assays with good selectivity over other nuclear hormone receptors.
| Price | 992,00 RON (preturile sunt fara TVA) |
|---|---|
| Description |
Brilanestrant (GDC-0810, ARN-810） is a potent ER-αbinder (ER-α, IC50 = 6.1 nM; ER-β, IC50 = 8.8 nM), a full transcriptional antagonist with no agonism and displays good potency and efficacy in ER-α degradation (EC50 = 0.7 nM) and MCF-7 breast cancer cell viability (IC50 = 2.5 nM) assays with good selectivity over other nuclear hormone receptors. |
